Buy Dechloroetizolam Pellets 5mg Online | High-Purity Thienotriazolodiazepine Research Chemical
Introduction to Buy Dechloroetizolam Pellets 5mg
Buy Dechloroetizolam Pellets 5mg (2-deschloroetizolam), designated in pharmacological and forensic literature as a novel synthetic thienotriazolodiazepine, is a highly potent research chemical and a critical reference standard in neuropharmacological and forensic toxicology research. Structurally, it is the direct 2-deschloro analog of the well-documented etizolam, lacking the chlorine atom at the 2-position of the phenyl ring.
Crucially, Dechloroetizolam is not merely a structural analog; it is the primary active metabolite of etizolam, formed via hepatic oxidative dechlorination. In neuropharmacological research, Dechloroetizolam functions as a positive allosteric modulator (PAM) at the GABA_A receptor, exhibiting high affinity and efficacy. Because it is the metabolite that actually exerts prolonged receptor occupancy after etizolam ingestion, it is indispensable for pharmacokinetic modeling. Because handling bulk thienotriazolodiazepine powders poses severe risks of accidental exposure and dosing errors, we supply Dechloroetizolam in precision-dosed 5mg pressed pellets. This format guarantees absolute dosing accuracy, eliminates the hazards associated with loose powders, and provides a highly convenient metric for streamlined volumetric preparation (e.g., dissolving one 5mg pellet in 5mL of solvent yields an exact 1mg/mL standard). Note: This product is strictly intended for in-vitro research and analytical purposes only.
Key Features and Benefits – Buy Dechloroetizolam Pellets 5mg
- Absolute Dosing Precision: Each pellet contains exactly 5mg of Dechloroetizolam, eliminating the life-threatening risk of micro-weighing errors inherent with active bulk powders and ensuring absolute consistency across your research assays.
- Streamlined Volumetric Preparation: The 5mg metric provides a highly convenient, standardized reference mass for easy mathematical dilution (e.g., yielding exactly 1mg/mL in 5mL, or 0.1mg/mL in 50mL) without the fractional calculations required by random bulk powder masses.
- Active Metabolite Modeling: Provides researchers with the direct active metabolite of etizolam, essential for mapping the pharmacokinetic pathways, metabolic clearance, and prolonged receptor occupancy of thienotriazolodiazepines.
- Halogen-Removal SAR Mapping: Dechloroetizolam provides researchers with a vital tool to study the structural-activity relationships (SAR) of halogenated vs. non-halogenated diazepines, isolating how the removal of the 2-chloro group alters receptor subunit selectivity and binding kinetics.
- Enhanced Laboratory Safety: The pressed pellet format drastically reduces the risk of accidental aerial dispersion or transdermal absorption, which is a severe hazard with loose, potent benzodiazepine powders.
Product Specifications
- Chemical Name: 2-ethyl-9-methyl-6-phenyl-4H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine
- Common Designation: Dechloroetizolam / 2-Deschloroetizolam
- CAS Number: Refer to Certificate of Analysis
- Class: Thienotriazolodiazepine / GABA_A PAM / Research Chemical
- Dosage per Unit: 5 mg (Precisely measured and pressed)
- Format: Pressed pellets in tamper-evident, light-resistant packaging
- Purity: ≥ 98% (Verified by Independent Third-Party Testing)
- Appearance: White to off-white pressed solid pellets (shape/color varies by batch)
- Storage Requirements: Store in a cool, dry, dark environment (ideally -20°C for long-term archival). Keep in original packaging to protect from light and humidity.
- Solubility: Freely soluble in DMSO, ethanol, and slightly soluble in warm aqueous buffers once extracted from the pellet matrix.
Applications and Usage
Dechloroetizolam 5mg Pellets are exclusively designated for in-vitro (outside a living organism) research and analytical applications. Common laboratory applications include:
- Volumetric Standard Preparation: Utilizing the exact 5mg metric to create large-volume, precisely concentrated stock solutions for high-throughput screening and sub-micromolar assay preparation.
- Metabolite Pharmacokinetic Profiling: Utilizing Dechloroetizolam as a reference standard to map the metabolic clearance, half-life, and accumulation potential of the primary active metabolite of etizolam in hepatocyte and blood plasma models.
- GABA_A Receptor Binding Assays: Investigating the compound’s affinity and efficacy as a positive allosteric modulator at the benzodiazepine binding site on GABA_A receptors, comparing its binding kinetics to its parent compound (etizolam).
- Halogen-Removal SAR Studies: Contrasting the pharmacokinetic properties and receptor conformational changes induced by the removal of the 2-chloro group versus the halogenated core to isolate how halogens dictate thienotriazolodiazepine potency.
- Forensic Toxicology Calibration: Utilizing the precisely dosed 5mg pellet as a known quantitative standard for LC/MS and GC/MS spectroscopy to validate analytical instruments, establish limits of detection, and confirm etizolam ingestion via metabolite detection in biological matrices.
Disclaimer: This product is not for human or veterinary consumption. It must only be handled in controlled laboratory environments by qualified professionals.
Purity and Testing
We guarantee a purity level of ≥ 98% for the Dechloroetizolam utilized in our pellets. Every production batch undergoes rigorous, independent third-party testing to verify chemical identity, absolute purity, dosage accuracy, and the absence of dangerous residual solvents, heavy metals, or unreacted precursors. Because benzodiazepines are a highly regulated and counterfeited class, we perform exhaustive screening to ensure the absolute absence of dangerous substituted benzodiazepine contaminants (such as etizolam, flualprazolam, or flubromazolam). Certificates of Analysis (CoA) and Safety Data Sheets (SDS) are provided upon request.
Safety and Handling
WARNING: DECHLOROETIZOLAM IS A HIGHLY POTENT CENTRAL NERVOUS SYSTEM DEPRESSANT. EXTREME CAUTION IS REQUIRED.
- Personal Protective Equipment (PPE): Must wear nitrile gloves, chemical-resistant safety goggles, and a P100 particulate respirator when handling the pellets or extracting the compound.
- Extraction Safety: When crushing or dissolving the 5mg pellet to extract the dose for assays, do so within a certified chemical fume hood using appropriate non-sparking tools.
- Accidental Exposure: If skin contact occurs, wash thoroughly with soap and water immediately. Seek medical attention if physiological effects occur. Note: Opioid antagonists like Naloxone are generally ineffective against benzodiazepine toxicity; flumazenil is the specific antagonist, but may precipitate seizures.
- Secure Storage: Keep pellets locked away in a secure, access-controlled laboratory cabinet, out of reach of unauthorized personnel.
Global Shipping and Discreet Delivery
- Global Reach: We ship Dechloroetizolam Pellets internationally, complying with all hazardous materials shipping regulations.
- Discreet Packaging: Orders are dispatched in unmarked, tamper-evident packaging. The uniform shape of supplement bottles makes them exceptionally easy to ship discreetly without attracting unwanted attention.
- Rapid Processing: Orders are processed and shipped within 24 hours of cleared payment with full end-to-end tracking.
- Damage Prevention: Pellet containers are cushioned within rigid outer boxes to prevent crushing during international transit.
Why Choose Us To Buy Dechloroetizolam Pellets 5mg?
- Innovative Delivery Formats: We are pioneers in providing high-potency research chemicals in precision-dosed, laboratory-friendly formats that prioritize safety and volumetric accuracy over dangerous bulk powders.
- Uncompromising Quality: We verify every batch in-house and via third-party labs—including exhaustive contaminant screening—before it reaches you.
- Total Transparency: Full analytical data provided—no fillers, no impurities, just verified 5mg reference units.
- Secure Transactions: We utilize SSL encryption and accept secure, discreet payment methods, including major cryptocurrencies (Bitcoin, Monero, Ethereum) and secure bank transfers.
Legal and Safety Compliance
Dechloroetizolam 5mg Pellets are sold strictly as research chemicals and are not approved by the FDA, EMA, or any equivalent regulatory body for human or veterinary use.
It is the sole responsibility of the purchaser to ensure that the acquisition, possession, and use of Dechloroetizolam comply with all local, state, national, and international laws. Warning: Dechloroetizolam is a potent central nervous system depressant and GABA_A agonist. Ingestion can cause severe, life-threatening psychological and physiological effects, including profound sedation, respiratory depression, coma, and death. As the primary active metabolite of etizolam, it may fall under federal analogue acts or specific benzodiazepine/NPS legislation in various jurisdictions. We do not ship to regions where this compound is explicitly prohibited. By purchasing from us, you affirm that you are a qualified researcher or institutional buyer over the age of 18, and you assume all legal liability for the product upon delivery.
Frequently Asked Questions (FAQ)
Q1: What is Dechloroetizolam?
A: Dechloroetizolam (2-deschloroetizolam) is a synthetic thienotriazolodiazepine. It acts as a positive allosteric modulator at the GABA_A receptor. Crucially, it is the primary active metabolite of etizolam, meaning it is the chemical compound that remains after the body enzymatically removes the chlorine atom from etizolam.
Q2: Why choose 5mg pellets over bulk Dechloroetizolam powder?
A: The 5mg pressed pellet guarantees an exact, pre-measured reference mass, removing the risk of micro-weighing errors associated with potent bulk powders. The specific 5mg metric is highly optimized for streamlined volumetric dilution—dissolving one pellet in 5mL of solvent instantly creates an exact 1mg/mL solution, eliminating complex fractional math and saving significant laboratory preparation time.
Q3: What makes Dechloroetizolam different from Etizolam?
A: Structurally, Dechloroetizolam lacks the 2-chloro group found on the phenyl ring of Etizolam. Pharmacologically, Dechloroetizolam is the active metabolite of Etizolam. This provides a vital tool for comparative SAR (Structural-Activity Relationship) research, allowing researchers to isolate how the removal of the halogen alters receptor binding kinetics and metabolic clearance.
Q4: Can the contents of the pellet be consumed?
A: Absolutely NOT. Dechloroetizolam is a potent CNS depressant. Ingestion can cause profound, long-lasting sedation, respiratory depression, and death. It is strictly for in-vitro laboratory and analytical research and is strictly prohibited for human consumption.
Q5: Do you provide a Certificate of Analysis (CoA)?
A: Yes. We provide a comprehensive CoA—including HPLC, GC/MS, and dosage verification data—for every pellet batch we sell. This guarantees the identity, purity, and exact 5mg mass of the compound.
Q6: Is it legal to buy Dechloroetizolam in my country?
A: Legality varies drastically. Because it is the active metabolite of a scheduled benzodiazepine (Etizolam), it is often controlled under analogue acts or specific NPS bans. We cannot provide legal advice. It is your responsibility to research your local laws regarding this compound before placing an order.
Q7: How should I store Dechloroetizolam Pellets for long-term research?
A: Store the pellets in their original, tightly sealed container in a cool, dry, dark place (room temperature is typically sufficient, or 4°C for long-term storage). Keep away from direct sunlight, heat, and moisture to prevent degradation of the active ingredient.




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